TY - JOUR
T1 - Synthesis of some secondary amine derivatives bearing a heteroaryl fragment
AU - Kouznetsov, Vladímir V.
AU - Saavedra, Luis Astudillo
AU - Vargas Méndeź, Leonor Y.
AU - Cazar Ramírez, Maria E.
PY - 2004/12
Y1 - 2004/12
N2 - Diverse N-(heteroarylmethyl)anilines were easily prepared from corresponding aldimines derived from commercially available aromatic aldehydes and anilines. New series of substituted NH-tetrahydroquinolines were also prepared using imino-Diels-Alder reaction between aldimines and N-vinylpyrrolidin-2-one in the presence of BF3OEt2 and the multi-component condensation reactions using a friendly ecological catalyst (BiCl3). The secondary amines obtained bearing a heteroaryl moiety were tested as possible antibacterial and antifungal agents.
AB - Diverse N-(heteroarylmethyl)anilines were easily prepared from corresponding aldimines derived from commercially available aromatic aldehydes and anilines. New series of substituted NH-tetrahydroquinolines were also prepared using imino-Diels-Alder reaction between aldimines and N-vinylpyrrolidin-2-one in the presence of BF3OEt2 and the multi-component condensation reactions using a friendly ecological catalyst (BiCl3). The secondary amines obtained bearing a heteroaryl moiety were tested as possible antibacterial and antifungal agents.
UR - https://www.scopus.com/pages/publications/13244277681
U2 - 10.4067/s0717-97072004000400010
DO - 10.4067/s0717-97072004000400010
M3 - Artículo
AN - SCOPUS:13244277681
SN - 0717-9324
VL - 49
SP - 319
EP - 325
JO - Journal of the Chilean Chemical Society
JF - Journal of the Chilean Chemical Society
IS - 4
ER -